Please use this identifier to cite or link to this item:
https://hdl.handle.net/11147/10233
Title: | 1,2-Diborolanes with strong donor substituents: Synthesis and high antimicrobial activity | Authors: | Şahin, Yüksel Poyrazoğlu Çoban, Esin Sevinçek, Resul Bıyık, Halil H. Özgener, Hüseyin Aygün, Muhittin |
Keywords: | Antimicrobial Diboracyclopentane Diborolane Heterocycles |
Issue Date: | 2021 | Publisher: | Academic Press | Abstract: | 1,2-diborolanes with strong and without strong donor substituents have been described, and are also referred to as 1,2-diboracyclopentane. The 1,2-diaryl/alkyl-amino-1,2-diboracyclopentanes 2, 3, and 4 were obtained in good yield after the reaction of 1,2-dichloro-1,2-diboracyclopentane 1 with ArNHLi and Me3Si-NR2. The structures of these new derivatives were characterized by nuclear magnetic resonance spectroscopy. The molecular structures of 2b, 2c, 2e, 4, and 5f were also determined by single-crystal X-ray diffraction. The newly synthesized 1,2-borolanes are stable in air and showed particularly high activity against some Gram-positive bacteria. © 2020 Elsevier Inc. | URI: | https://doi.org/10.1016/j.bioorg.2020.104494 https://hdl.handle.net/10233 |
ISSN: | 0045-2068 1090-2120 |
Appears in Collections: | Chemistry / Kimya PubMed İndeksli Yayınlar Koleksiyonu / PubMed Indexed Publications Collection Scopus İndeksli Yayınlar Koleksiyonu / Scopus Indexed Publications Collection WoS İndeksli Yayınlar Koleksiyonu / WoS Indexed Publications Collection |
Files in This Item:
File | Size | Format | |
---|---|---|---|
1-s2.0-S0045206820317922-main.pdf Until 2024-01-01 | 1.63 MB | Adobe PDF | View/Open Request a copy |
CORE Recommender
SCOPUSTM
Citations
4
checked on Dec 9, 2023
WEB OF SCIENCETM
Citations
1
checked on Jun 17, 2023
Page view(s)
34
checked on Dec 11, 2023
Google ScholarTM
Check
Altmetric
Items in GCRIS Repository are protected by copyright, with all rights reserved, unless otherwise indicated.