Please use this identifier to cite or link to this item:
|Title:||1,2-Diborolanes with strong donor substituents: Synthesis and high antimicrobial activity||Authors:||Şahin, Yüksel
Poyrazoğlu Çoban, Esin
Bıyık, Halil H.
|Issue Date:||2020||Publisher:||Academic Press Inc.||Abstract:||1,2-diborolanes with strong and without strong donor substituents have been described, and are also referred to as 1,2-diboracyclopentane. The 1,2-diaryl/alkyl-amino-1,2-diboracyclopentanes 2, 3, and 4 were obtained in good yield after the reaction of 1,2-dichloro-1,2-diboracyclopentane 1 with ArNHLi and Me3Si-NR2. The structures of these new derivatives were characterized by nuclear magnetic resonance spectroscopy. The molecular structures of 2b, 2c, 2e, 4, and 5f were also determined by single-crystal X-ray diffraction. The newly synthesized 1,2-borolanes are stable in air and showed particularly high activity against some Gram-positive bacteria. © 2020 Elsevier Inc.||URI:||https://doi.org/10.1016/j.bioorg.2020.104494
|Appears in Collections:||Scopus İndeksli Yayınlar Koleksiyonu / Scopus Indexed Publications Collection|
Show full item record
checked on Dec 8, 2021
Items in GCRIS Repository are protected by copyright, with all rights reserved, unless otherwise indicated.